I-ActiTide™ AH3 / Acetyl Hexapeptide-8

Incazelo emfushane:

I-ActiTide™ AH3 iyisiqeshana se-hexapeptide esilingisa isakhiwo seprotheyini ye-SNAP-25. Incintisana ne-SNAP-25, ivimbela ukwakheka kwe-SNARE complex ene-syntaxin kanye ne-VAMP. Lokhu kuvinjelwa kuvimbela ukuhlangana kwe-membrane kanye nokukhululwa okulandelayo kwama-neurotransmitters. Njengesithako esinciphisa imibimbi ngokushesha, i-ActiTide™ AH3 inciphisa ngempumelelo imibimbi enamandla ebangelwa ukufinyela kwemisipha endaweni futhi isiza ukunciphisa inani kanye nokujula kwemigqa yokuveza. Ngaphezu kwalokho, imnene, ayinabo ubuthi, futhi ifanele zonke izinhlobo zesikhumba. I-ActiTide™ AH3 isetshenziswa kabanzi emikhiqizweni yobuhle kanye nokunakekelwa kwesikhumba, kufaka phakathi ama-serum okulwa nemibimbi, okhilimu bobuso, okhilimu bamehlo, izimonyo eziyisisekelo, kanye namamaski, okunikeza izinzuzo eziphelele zokulwa nokuguga.


Imininingwane Yomkhiqizo

Amathegi Omkhiqizo

I gama le-brand I-ActiTide™ AH3
Inombolo ye-CAS 616204-22-9
Igama le-INCI I-Acetyl Hexapeptide-8
Isicelo Iloshini, Ama-Serum, Imaski, Isihlanzi Sobuso
Iphakheji 100g/ibhodlela, 1kg/isikhwama
Ukubukeka Impuphu emhlophe kuya kwemhlophe kakhulu
Ukuncibilika Amanzi ancibilikayo
Umsebenzi Uchungechunge lwe-Peptide
Isikhathi sokuphelelwa yisikhathi iminyaka engu-2
Isitoreji Gcina isitsha sivalwe kahle endaweni epholile, eyomile ku-2 - 8°C.
Isilinganiso 0.005-0.05%

Isicelo

 

Ucwaningo ngezindlela eziyisisekelo zokulwa nemibimbi luholele ekutholakaleni kwe-ActiTide™ AH3, i-hexapeptide entsha eyathuthukiswa ngendlela yesayensi kusukela ekwakhiweni okunengqondo kuya ekukhiqizweni kwe-GMP, kwaba nemiphumela emihle.

I-ActiTide™ AH3 inikeza ukusebenza kahle kokunciphisa imibimbi okufana nohlobo lwe-Botulinum Toxin A, ngenkathi igwema izingozi zomjovo futhi inikeza ukusebenza kahle okukhulu kwezindleko.

 

Izinzuzo Zobuhle:

I-ActiTide™ AH3 yehlisa ukujula kwemibimbi okubangelwa ukufinyela kwemisipha yobuso, okunemiphumela evelele ebunzini kanye nemibimbi ye-periocular.

 

Indlela Yokusebenza:

Ukufinyela kwemisipha kwenzeka lapho kukhululwa i-neurotransmitter kuma-vesicle e-synaptic. I-SNARE complex – i-ternary assembly yama-protein e-VAMP, i-Syntaxin, ne-SNAP-25 – ibalulekile ekubekweni kwe-vesicle kanye ne-neurotransmitter exocytosis (A. Ferrer Montiel et al., JBC 1997, 272:2634-2638). Le complex isebenza njenge-hook yeselula, ibamba ama-vesicle futhi iqhube ukuhlangana kwe-membrane.

Njengokulingisa kwesakhiwo se-SNAP-25 N-terminus, i-ActiTide™ AH3 incintisana ne-SNAP-25 ukuze ifakwe ku-SNARE complex, iguqula ukuhlanganiswa kwayo. Ukuwohloka kwe-SNARE complex kuphazamisa ukugoba kwe-vesicle kanye nokukhululwa kwe-neurotransmitter okulandelayo, okuholela ekunciphiseni ukufinyela kwemisipha kanye nokuvimbela ukwakheka kwemibimbi kanye nomugqa omncane.

I-ActiTide™ AH3 iyindlela ephephile, engabizi kakhulu, futhi ethambile esikhundleni se-Botulinum Toxin Type A. Ihlose ngqo indlela efanayo yokwakheka kwemibimbi kodwa isebenza ngendlela ehlukile.


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