I gama le-brand | I-ActiTide-AH3 |
Inombolo ye-CAS. | 616204-22-9 |
Igama le-INCI | I-Acetyl Hexapeptide-8 |
Isicelo | I-lotion, iSerum, Imaski, isihlanzi sobuso |
Iphakheji | 100g/ibhodlela, 1kg/isikhwama |
Ukubukeka | Impushana emhlophe ukuya kokumhlophe |
Ukuncibilika | Amanzi ancibilikayo |
Umsebenzi | Peptide series |
Impilo yeshelufu | iminyaka engu-2 |
Isitoreji | Gcina isitsha sivalwe ngokuqinile endaweni epholile, eyomile eku-2 - 8°C. |
Umthamo | 0.005-0.05% |
Isicelo
Ucwaningo lwezindlela eziyisisekelo zokunqanda imibimbi luholele ekutholweni kwe-ActiTide-AH3, i-hexapeptide esungulwe ngendlela yesayensi ukusuka kumklamo ophusile kuya ekukhiqizweni kwe-GMP, kube nemiphumela emihle.
I-ActiTide-AH3 iletha ukusebenza ngempumelelo kokunciphisa imibimbi okuqhathaniswa nohlobo A lwe-Botulinum Toxin, kuyilapho igwema izingozi zokujova futhi inikeza ukusebenza kahle kwezindleko.
Izinzuzo Zezimonyo:
I-ActiTide-AH3 yehlisa ukujula kokushwabana okubangelwa ukufinyela kwemisipha yobuso, ibe nemiphumela evelele ebunzini kanye nemibimbi ye-periocular.
Indlela Yesenzo:
Ukufinyela kwemisipha kwenzeka lapho i-neurotransmitter ikhishwa kuma-synaptic vesicles. I-SNARE complex - i-ternary assembly yamaprotheni e-VAMP, i-Syntaxin, ne-SNAP-25 - ibalulekile ku-vesicle docking kanye ne-neurotransmitter exocytosis (A. Ferrer Montiel et al., JBC 1997, 272: 2634-2638). Le nkimbinkimbi isebenza njengehuku lamaselula, ibamba ama-vesicles futhi iqhube ukuhlanganiswa kwe-membrane.
Njenge-mimetic yesakhiwo ye-SNAP-25 N-terminus, i-ActiTide-AH3 incintisana ne-SNAP-25 ukuze ifakwe kunxanxathela ye-SNARE, imodela ukuhlanganiswa kwayo. Ukungaqini kahle kwenkimbinkimbi ye-SNARE kukhubaza ukudotshwa kwe-vesicle kanye nokukhululwa kwe-neurotransmitter okulandelayo, okuholela ekunciphiseni ukufinyela kwemisipha kanye nokuvimbela ukushwabana nokwakheka komugqa omuhle.
I-ActiTide-AH3 iyindlela ephephile, eyonga kakhulu, futhi emnene kune-Botulinum Toxin Type A. Iqondise ngokuqondile indlela efanayo yokwenza imibimbi kodwa isebenza ngendlela ehlukile.