I-ActiTide™ AH3 / Acetyl Hexapeptide-8

Incazelo emfushane:

I-ActiTide™ AH3 iwucezu lwe-hexapeptide elingisa isizinda sesakhiwo sephrotheni ye-SNAP-25. Iqhudelana ne-SNAP-25, ivimbela ukwakheka kwe-SNARE complex ne-syntaxin ne-VAMP. Lokhu kuvinjelwa kuvimbela ukuhlanganiswa kwe-membrane kanye nokukhululwa okulandelayo kwama-neurotransmitters. Njengesithako esinciphisa ukushwabana ngokushesha, i-ActiTide™ AH3 inciphisa ngempumelelo imibimbi eguquguqukayo ebangelwa ukufinyela kwemisipha yendawo futhi isiza ukwehlisa inombolo nokujula kwemigqa yokukhuluma. Ngaphezu kwalokho, imnene, ayinabo ubuthi, futhi ifanele zonke izinhlobo zesikhumba. I-ActiTide™ AH3 isetshenziswa kakhulu emikhiqizweni yobuhle ne-skincare, okuhlanganisa ama-serum aqeda imibimbi, okhilimu bobuso, okhilimu wamehlo, izimonyo eziyisisekelo, namamaski, anikeza izinzuzo ezibanzi zokulwa nokuguga.


Imininingwane Yomkhiqizo

Omaka bomkhiqizo

I gama le-brand I-ActiTide™ AH3
Inombolo ye-CAS. 616204-22-9
Igama le-INCI I-Acetyl Hexapeptide-8
Isicelo I-Lotion, iSerum, Imaski, Isihlanzi sobuso
Iphakheji 100g/ibhodlela, 1kg/isikhwama
Ukubukeka Impushana emhlophe ukuya kokumhlophe
Ukuncibilika Amanzi ancibilikayo
Umsebenzi Peptide series
Impilo yeshelufu iminyaka engu-2
Isitoreji Gcina isitsha sivalwe ngokuqinile endaweni epholile, eyomile eku-2 - 8°C.
Umthamo 0.005-0.05%

Isicelo

 

Ucwaningo lwezindlela eziyisisekelo zokunqanda imibimbi luholele ekutholweni kwe-ActiTide™ AH3, i-hexapeptide esungulwe ngendlela yesayensi ukusuka kumklamo ophusile kuya ekukhiqizweni kwe-GMP, kube nemiphumela emihle.

I-ActiTide™ AH3 iletha ukusebenza ngempumelelo kokunciphisa imibimbi okuqhathaniswa nohlobo A lwe-Botulinum Toxin, kuyilapho igwema izingozi zokujova futhi inikeza ukusebenza ngempumelelo kwezindleko.

 

Izinzuzo Zezimonyo:

I-ActiTide™ AH3 yehlisa ukujula kokushwabana okubangelwa ukufinyela kwemisipha yobuso, ibe nemiphumela ezwakalayo ebunzini kanye nemibimbi ye-periocular.

 

Indlela Yesenzo:

Ukufinyela kwemisipha kwenzeka lapho kukhululwa i-neurotransmitter kuma-synaptic vesicles. I-SNARE complex - i-ternary assembly yamaprotheni e-VAMP, i-Syntaxin, ne-SNAP-25 - ibalulekile ku-vesicle docking kanye ne-neurotransmitter exocytosis (A. Ferrer Montiel et al., JBC 1997, 272: 2634-2638). Le nkimbinkimbi isebenza njengehhuku yeselula, ibamba ama-vesicles futhi iqhube ukuhlanganiswa kwe-membrane.

Njenge-mimetic yesakhiwo ye-SNAP-25 N-terminus, i-ActiTide™ AH3 incintisana ne-SNAP-25 ukuze ifakwe kunxanxathela ye-SNARE, imodela ukuhlanganiswa kwayo. Ukungaqini kahle kwenkimbinkimbi ye-SNARE kukhubaza ukudotshwa kwe-vesicle kanye nokukhululwa kwe-neurotransmitter okulandelayo, okuholela ekunciphiseni ukufinyela kwemisipha kanye nokuvimbela ukushwabana nokwakheka komugqa omuhle.

I-ActiTide™ AH3 iyindlela ephephile, eyonga kakhulu, futhi emnene kune-Botulinum Toxin Type A. Iqondise ngokuqondile indlela efanayo yokushwabana kodwa isebenza ngendlela ehlukile.


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