I-ActiTide™ PT7 / Palmitoyl Tetrapeptide-7

Incazelo emfushane:

I-Immunoglobulin G (IgG) iyisakhi esiyinhloko sama-immunoglobulin egazini lomuntu kanye ne-antibody eningi kakhulu emzimbeni. I-ActiTide™ PT7 iyi-palmitoylated derivative ye-Gly-Gln-Pro-Arg (GQPR) tetrapeptide, etholakala ku-structural fragment (341-344) ye-immunoglobulin G heavy chain. Izifundo zibonise ukuthi i-GQPR tetrapeptide ingavuselela ama-macrophage nama-neutrophils, ithuthukise umsebenzi we-phagocytic. Ngaphezu kwalokho, i-GQP iwuchungechunge oluvamile lwe-tripeptide olutholakala ku-type IV collagen. Njenge-ejenti yokulungisa isikhumba, i-ActiTide™ PT7 ingavimbela ukukhiqizwa kwama-cytokines okuvuvukala (IL-6), ikhuthaze ukwakheka kwe-laminin, i-fibronectin, kanye ne-collagen, inciphise imibimbi yesikhumba, futhi inemiphumela eduduzayo neqinisayo.


Imininingwane Yomkhiqizo

Amathegi Omkhiqizo

I gama le-brand I-ActiTide™ PT7
Inombolo ye-CAS 221227-05-0
Igama le-INCI I-Palmitoyl Tetrapeptide-7
Isicelo Iloshini, Ama-Serum, Imaski, Isihlanzi Sobuso
Iphakheji 100g/ibhodlela
Ukubukeka Impuphu emhlophe kuya kwemhlophe kakhulu
Ukuncibilika Ayincibiliki emanzini
Umsebenzi Uchungechunge lwe-Peptide
Isikhathi sokuphelelwa yisikhathi iminyaka engu-2
Isitoreji Gcina isitsha sivalwe kahle endaweni epholile, eyomile ku-2 - 8°C.
Isilinganiso 0.001-0.1% ngaphansi kwama-45 °C

Isicelo

 

I-ActiTide™ PT7 iyi-peptide esebenzayo elingisa ingxenye ye-immunoglobulin IgG. Iguqulwe nge-palmitoylation, ikhombisa ukuzinza okuthuthukisiwe kanye namandla okumunca i-transdermal, okwenza kube lula ukungena esikhumbeni ngempumelelo ukuze isebenze kahle.

 

Indlela Eyinhloko Yokusebenza: Ukulawula Ukuvuvukala

Isici Esiyinhloko Sokuqondisa:

Indlela yayo eyinhloko isekunciphiseni kakhulu ukukhiqizwa kwe-cytokine Interleukin-6 (IL-6) ekhuthaza ukuvuvukala.

Ukunciphisa Impendulo Yokuvuvukala:

I-IL-6 ingumlamuleli obalulekile ezinqubweni zokuvuvukala kwesikhumba. Ukugxila okuphezulu kwe-IL-6 kubhebhethekisa ukuvuvukala, kusheshise ukuwohloka kwe-collagen namanye amaprotheni abalulekile esikhumba, ngaleyo ndlela kukhuthaze ukuguga kwesikhumba. I-Palmitoyl Tetrapeptide-7 isebenza kuma-keratinocyte esikhumba kanye nama-fibroblast ngokukhuthaza isignali, ilawula izimpendulo zokuvuvukala, ikakhulukazi ngokuvimbela ukukhishwa ngokweqile kwe-IL-6 emangqamuzaneni amhlophe egazi.

Ukuvinjelwa Okuxhomeke Kumthamo:

Izifundo zelebhu ziqinisekisa ukuthi ivimbela ukukhiqizwa kwe-IL-6 ngendlela encike kumthamo; amazinga aphezulu aveza imiphumela ebaluleke kakhulu yokuvimbela (kufika ku-40% izinga eliphezulu lokuvimbela).

Isebenza Kakhulu Ekulimaleni Kwesithombe:

Ezimweni lapho imisebe ye-ultraviolet (UV) ibangela ukukhiqizwa okukhulu kwe-IL-6, amaseli aphathwe nge-Palmitoyl Tetrapeptide-7 abonisa izinga lokuvinjelwa kokukhiqizwa kwe-IL-6 kufika ku-86%.

 

Ukusebenza Okuyinhloko kanye Nezinzuzo:

Kuthulisa Futhi Kunciphise Ukuvuvukala:

Ngokuvimbela ngempumelelo izici zokuvuvukala njenge-IL-6, kunciphisa ukusabela okungafanele kokuvuvukala kwesikhumba, kunciphisa ukubomvu nokungakhululeki.

Kuvikela Ekulimaleni Kwemvelo:

Kusiza ukugcina ibhalansi yama-cytokine esikhumba, kuvikela isikhumba ekulimaleni kwemvelo (njengemisebe ye-UV) kanye nomonakalo we-glycation.

Kukhuthaza Ithoni Yesikhumba Elinganayo:

Ukunciphisa ukuvuvukala kusiza ukuthuthukisa ukubomvu kwesikhumba kanye nezinye izinkinga zethoni engalingani, okungenzeka kusize ekukhanyiseni ibala ukuze kube nethoni yesikhumba elinganayo.

Ukubambezeleka Izimpawu Zokuguga:

Ngokunciphisa ukuvuvukala nokuvimbela ukuwohloka kwe-collagen, kusiza ukulwa nezimpawu zokuguga ezifana nemibimbi nokuwa.

Ukuthuthukiswa Kokubambisana:

Uma ihlanganiswa nezinye izithako ezisebenzayo (njengePalmitoyl Tripeptide-1), isibonelo ku-Matrixyl 3000 complex, ikhiqiza imiphumela yokusebenzisana, ithuthukisa imiphumela yokulwa nokuguga iyonke.

 

Isicelo:

I-ActiTide-PT7 isetshenziswa kabanzi emikhiqizweni yokunakekelwa kwesikhumba, ikakhulukazi idlala indima ebalulekile ekulungiseni isikhumba, ekuthobeni ukuvuvukala, kanye nemikhiqizo yokuqinisa imibimbi.


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